Determine the necessary mass, volume, or concentration for preparing a solution.
Synonyms | R6238-d4-1 |
---|---|
Specifications & Purity | Moligand™, ≥95 atom% D,≥95% |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Grade | Moligand™ |
Product Description | Pimozide-d 4 -1 is the deuterium labeled Pimozide. Pimozide is a dopamine receptor antagonist , with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozid Appearance:Solid In Vitro:Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the phar Biological Activity:Pimozide-d 4 -1 is the deuterium labeled Pimozide. Pimozide is a dopamine receptor antagonist , with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozid |
Canonical SMILES | O=C1NC2=C([2H])C([2H])=C([2H])C([2H])=C2N1C3CCN(CCCC(C4=CC=C(F)C=C4)C5=CC=C(F)C=C5)CC3 |
---|---|
Alternate CAS | 2062-78-4(unlabelled) |
Molecular Weight | 465.57 |
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
---|---|---|---|
![]() | Certificate of Analysis | Oct 25, 2024 | P658709 |
Starting at $103.90