| SKU | Size | Availability | Price | Qty |
|---|---|---|---|---|
| U423533-1ml | 1ml | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $69.90 |
| Synonyms | urapidil | 34661-75-1 | Ebrantil | Eupressyl | Mediatensyl | Uraprene | 6-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]amino]-1,3-dimethyluracil | NSC 310405 | B-66256 | 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1,3-dimethylpyrimidine-2,4-dione | NSC-310405 | A78GF |
|---|---|
| Specifications & Purity | 10mM in DMSO |
| Storage Temp | Store at -80°C |
| Shipped In | Ice chest + Ice pads |
| Product Description | Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist. |
| Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
|---|
| IUPAC Name | 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1,3-dimethylpyrimidine-2,4-dione |
|---|---|
| INCHI | InChI=1S/C20H29N5O3/c1-22-18(15-19(26)23(2)20(22)27)21-9-6-10-24-11-13-25(14-12-24)16-7-4-5-8-17(16)28-3/h4-5,7-8,15,21H,6,9-14H2,1-3H3 |
| InChi Key | ICMGLRUYEQNHPF-UHFFFAOYSA-N |
| Canonical SMILES | CN1C(=CC(=O)N(C1=O)C)NCCCN2CCN(CC2)C3=CC=CC=C3OC |
| Isomeric SMILES | CN1C(=CC(=O)N(C1=O)C)NCCCN2CCN(CC2)C3=CC=CC=C3OC |
| RTECS | YQ9862000 |
| PubChem CID | 5639 |
| Molecular Weight | 387.48 |
| Reaxy-Rn | 725782 |
| Pictogram(s) | GHS07 |
|---|---|
| Signal | Warning |
| Hazard Statements | H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation H302:Harmful if swallowed |
| Precautionary Statements | P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing. P280:Wear protective gloves/protective clothing/eye protection/face protection. P302+P352:IF ON SKIN: wash with plenty of water. P321:Specific treatment (see ... on this label). P405:Store locked up. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P271:Use only outdoors or in a well-ventilated area. P270:Do not eat, drink or smoke when using this product. P304+P340:IF INHALED: Remove person to fresh air and keep comfortable for breathing. P403+P233:Store in a well-ventilated place. Keep container tightly closed. P362+P364:Take off contaminated clothing and wash it before reuse. P330:Rinse mouth. P264+P265:Wash hands [and …] thoroughly after handling. Do not touch eyes. P301+P317:IF SWALLOWED: Get medical help. P337+P317:If eye irritation persists: Get medical help. P332+P317:If skin irritation occurs: Get medical help. P319:Get medical help if you feel unwell. |
| RTECS | YQ9862000 |
| Reaxy-Rn | 725782 |
| Merck Index | 9865 |
| 1. Xinyi Yuan, Aerduosi Shayiranbieke, Ru Xu, Hongmei Jiang, Yushan Yang, Yajun Zhang, Guowei Yin, Xinfeng Zhao. (2022) Site-selective covalently immobilized alpha 1A adrenergic receptor for thermodynamic and extra-thermodynamic study of four ligands binding to the receptor by chromatographic methods. JOURNAL OF CHROMATOGRAPHY A, 1665 (462827). [PMID:35078002] [10.1016/j.chroma.2022.462827] |
| 2. Yanju Wu, Anxing Zhou, Huimin Yang, Fei Wang, Kui Lu. (2018) 3D Graphene-Nitrogen Doped Carbon Nanotubes Network Modified Electrode as Sensing Materials for the Determination of Urapidil. Materials, 11 (2): (322). [PMID:29473881] [10.3390/ma11020322] |
| 1. Xinyi Yuan, Aerduosi Shayiranbieke, Ru Xu, Hongmei Jiang, Yushan Yang, Yajun Zhang, Guowei Yin, Xinfeng Zhao. (2022) Site-selective covalently immobilized alpha 1A adrenergic receptor for thermodynamic and extra-thermodynamic study of four ligands binding to the receptor by chromatographic methods. JOURNAL OF CHROMATOGRAPHY A, 1665 (462827). [PMID:35078002] [10.1016/j.chroma.2022.462827] |
| 2. Yanju Wu, Anxing Zhou, Huimin Yang, Fei Wang, Kui Lu. (2018) 3D Graphene-Nitrogen Doped Carbon Nanotubes Network Modified Electrode as Sensing Materials for the Determination of Urapidil. Materials, 11 (2): (322). [PMID:29473881] [10.3390/ma11020322] |
