MS023 - 98%, high purity , CAS No.1831110-54-3, Inhibitor of coactivator associated arginine methyltransferase 1;Inhibitor of protein arginine methyltransferase 1;Inhibitor of protein arginine methyltransferase 3;Inhibitor of protein arginine methyltransferase 6;Inhibitor of protein arginine methyltran

Item Number

M275329

• Synonyms: N1-Methyl-N1-[[4-[4-(1-methylethoxy)phenyl]-1H-pyrrol-3-yl]methyl]-1,2-ethanediamine | N1-((4-(4-isopropoxyphenyl)-1H-pyrrol-3-yl)methyl)-N1-methylethane-1,2-diamine
• Specifications & Purity: Moligand™, ≥98%
• Biochemical and Physiological Mechanisms: MS023 is a potent, selective, and cell-active Type I PRMT inhibitor. IC 50 values are 30 nM (PRMT1), 119 nM (PRMT3), 83 nM (PRMT4), 4 nM (PRMT6) and 5 nM (PRMT8). It potently reduces cellular levels of H4R3me2a in MCF7 and HEK293 cells by inhibiting PRMT1
• Storage Temp: Store at -20°C
• Shipped In: Ice chest + Ice pads
• Grade: Moligand™
• Action Type: INHIBITOR
• Mechanism of action: Inhibitor of coactivator associated arginine methyltransferase 1;Inhibitor of protein arginine methyltransferase 1;Inhibitor of protein arginine methyltransferase 3;Inhibitor of protein arginine methyltransferase 6;Inhibitor of protein arginine methyltran
• Note: Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

Product Description

Shipped at 4°C. Store at -20°C.