GW 627368 - ≥98%(HPLC), high purity , CAS No.439288-66-1, Antagonist of EP 4 receptor

Item Number

G288949

Grouped product items
SKU	Size	Availability	Price
G288949-1mg	1mg	2	$15.90
G288949-5mg	5mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$64.90
G288949-10mg	10mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$97.90
G288949-25mg	25mg	2	$162.90
G288949-50mg	50mg	2	$271.90
G288949-250mg	250mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$1,224.90

Selective EP4receptor competitive antagonist

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Basic Description

Synonyms	A842355 \| NSC 96380 \| GW627368X \| GW-627368X \| BCP15277 \| CS-4458 \| EX-A603 \| GW 627368 \| SY029966 \| Benzeneacetamide, 4-(4,9-diethoxy-1,3-dihydro-1-oxo-2H-benz(f)isoindol-2-yl)-N-(phenylsulfonyl)- \| DB08074 \| HMS3650M04 \| 2-(4-(4,9-diethoxy-1-oxo-1,3-dih
Specifications & Purity	Moligand™, ≥98%(HPLC)
Biochemical and Physiological Mechanisms	Selective prostanoid EP4receptor competitive antagonist with additional affinity at TP receptors (pKivalues are 7.0 and 6.8 in competition radioligand bioassays). Affinity for all other prostanoid receptors is < 5.3. Inhibits U-46619 induced human platel
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of EP 4 receptor

Names and Identifiers

Pubchem Sid	504763559
Pubchem Sid Url	https://pubchem.ncbi.nlm.nih.gov/substance/504763559
IUPAC Name	N-(benzenesulfonyl)-2-[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]acetamide
INCHI	InChI=1S/C30H28N2O6S/c1-3-37-28-23-12-8-9-13-24(23)29(38-4-2)27-25(28)19-32(30(27)34)21-16-14-20(15-17-21)18-26(33)31-39(35,36)22-10-6-5-7-11-22/h5-17H,3-4,18-19H2,1-2H3,(H,31,33)
InChi Key	XREWXJVMYAXCJV-UHFFFAOYSA-N
Canonical SMILES	CCOC1=C2CN(C(=O)C2=C(C3=CC=CC=C31)OCC)C4=CC=C(C=C4)CC(=O)NS(=O)(=O)C5=CC=CC=C5
Isomeric SMILES	CCOC1=C2CN(C(=O)C2=C(C3=CC=CC=C31)OCC)C4=CC=C(C=C4)CC(=O)NS(=O)(=O)C5=CC=CC=C5
PubChem CID	5312130
Molecular Weight	544.62

Certificates（CoA,COO,BSE/TSE and Analysis Chart)

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7 results found

Lot Number	Certificate Type	Date	Item
L2412370	Certificate of Analysis	Dec 18, 2024	G288949
J2115201	Certificate of Analysis	Jul 15, 2024	G288949
J2115223	Certificate of Analysis	Jul 15, 2024	G288949
J2115247	Certificate of Analysis	Jul 15, 2024	G288949
J2115314	Certificate of Analysis	Jul 15, 2024	G288949
J2115348	Certificate of Analysis	Jul 15, 2024	G288949
J2115351	Certificate of Analysis	Jul 15, 2024	G288949

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Basic Description