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GSK 264220A - ≥98%(HPLC), high purity , CAS No.685506-42-7, Inhibitor of lipase G; endothelial type

GSK 264220A - ≥98%(HPLC), high purity , CAS No.685506-42-7, Inhibitor of lipase G; endothelial type

Item Number

G288505

Grouped product items
SKU	Size	Availability	Price	Qty
G288505-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$172.90
G288505-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$728.90

Endothelial lipase and lipoprotein lipase inhibitor

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Basic Description

Synonyms	N-[2-Methyl-5-(1-piperidinylsulfonyl)-3-furanyl]-N'-phenylurea \| 3-[2-methyl-5-(piperidine-1-sulfonyl)furan-3-yl]-1-phenylurea \| DTXSID30384608 \| HMS2799K10 \| Q27077890 \| SR-01000774442 \| CCG-242835 \| NCGC00344077-02 \| SMR000456118 \| HY-103372 \| GTPL6697
Specifications & Purity	Moligand™, ≥98%(HPLC)
Biochemical and Physiological Mechanisms	Endothelial lipase and lipoprotein lipase inhibitor (IC50values are 0.13 and 0.10μM respectively).
Storage Temp	Store at 2-8°C
Shipped In	Wet ice
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of lipase G; endothelial type

Mechanism of Action	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	References

IUPAC Name	1-(2-methyl-5-piperidin-1-ylsulfonylfuran-3-yl)-3-phenylurea
INCHI	InChI=1S/C17H21N3O4S/c1-13-15(19-17(21)18-14-8-4-2-5-9-14)12-16(24-13)25(22,23)20-10-6-3-7-11-20/h2,4-5,8-9,12H,3,6-7,10-11H2,1H3,(H2,18,19,21)
InChi Key	LVOVQRPAMXCXTM-UHFFFAOYSA-N
Canonical SMILES	CC1=C(C=C(O1)S(=O)(=O)N2CCCCC2)NC(=O)NC3=CC=CC=C3
Isomeric SMILES	CC1=C(C=C(O1)S(=O)(=O)N2CCCCC2)NC(=O)NC3=CC=CC=C3
PubChem CID	2810413
Molecular Weight	363.43

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